|
|
Name
|
Alternate Name
|
CAS Number
|
Catalog Number
|
Indication
|
| 1.
|
(+/-) KI-20227
|
Not Applicable
|
No CAS
|
KI-00590
|
Bone matastasis
|
| 2.
|
(+)-Tyrphostin B44
|
See Product Details
|
133550-37-5
|
KI-0483
|
See Product Details
|
| 3.
|
(R-) BL-2536
|
Not Applicable
|
No CAS
|
KI-00588
|
Thromboembolic disease
|
| 4.
|
(S-) BL-2536
|
Not Applicable
|
No CAS
|
KI-00587
|
Thromboembolic disease
|
| 5.
|
(S)-Roscovitine
|
See Product Details
|
186692-46-6
|
KI-0122
|
Cyclin-dependent kinase inhibitor
|
| 6.
|
1-Benzyl-3-Cetyl-2-Methylimidazolium Iodide
|
NH125
|
No CAS
|
KI-0504
|
CaM-Dependant Kinase III Inhibitor
|
| 7.
|
1H-Pyrazolo[3,4b]quinoxalin-3-amine
|
NSC 693868
|
40254-90-4
|
KI-0161
|
See Product Details
|
| 8.
|
4-(3-Pyridin-2-yl-1H-pyrazol-4-yl)-quinoline
|
LY-364947
|
396129-53-6
|
KI-0268
|
See Product Details
|
| 9.
|
4A-Phorbol 12,13-Dibutyrate
|
Not Applicable
|
93781-54-5
|
KI-0205
|
Protein kinase C inhibitor
|
| 10.
|
5,6-Dichlorobenzimidazole Riboside
|
DRB
|
53-85-0
|
KI-0129
|
CK2 (casein kinase-2) inhibitor
|
| 11.
|
5-iodotubercidin
|
Not Applicable
|
24386-93-4
|
KI-0177
|
Inhibitor of the enzyme adenosine kinase
|
| 12.
|
6-Dimethylaminopurine
|
Not Applicable
|
938-55-6
|
KI-0293
|
Protein kinase inhibitor
|
| 13.
|
7-hydroxy-1H-benzoimidazole
|
Not Applicable
|
No CAS
|
KI-00600
|
Alzheimer's disease
|
| 14.
|
A-134974
|
See Product Details
|
No CAS
|
KI-0437
|
Adenosine kinase (AK) inhibitor
|
| 15.
|
A-3 Hydrochloride
|
See Product Details
|
No CAS
|
KI-0241
|
Casein kinase (CK) inhibitor
|
| 16.
|
AB-1010
|
Mastinib
|
No CAS
|
KI-0294
|
TK inhibitor, selectively and effectively inhibiting c-kit
|
| 17.
|
ABT-737
|
Not Applicable
|
852808-04-9
|
KI-00579
|
Multiple myeloma
|
| 18.
|
ABT-869
|
Not Applicable
|
796967-16-3
|
KI-0438
|
Tyrosine kinase (RTK) inhibitor
|
| 19.
|
AC-220
|
Not Applicable
|
No CAS
|
KI-00601
|
Acute myeloid leukemia
|
| 20.
|
Aebsf Hydrochloride
|
4-(2-Aminoethyl)Benzene Sulfonyl Floride Hydrochloride
|
30827-99-7
|
KI-0490
|
See Product Details
|
| 21.
|
Aee-788
|
Not Applicable
|
No CAS
|
KI-0028
|
See Product Details
|
| 22.
|
AEG-33783
|
Not Applicable
|
No CAS
|
KI-0296
|
Inhibiting the JNK
|
| 23.
|
AEW-541
|
Not Applicable
|
No CAS
|
KI-0297
|
Kinase inhibitor of the IGF-IR
|
| 24.
|
AG 213
|
See Product Details
|
118409-60-2
|
KI-0298
|
See Product Details
|
| 25.
|
AG 494
|
Not Applicable
|
133550-35-3
|
KI-0300
|
Inhibitor of EGF receptor kinase
|
| 26.
|
AG 99
|
See Product Details
|
118409-59-9
|
KI-0303
|
See Product Details
|
| 27.
|
AG-1478
|
Not Applicable
|
153436-53-4
|
KI-0484
|
Tyrosine kinase inhibitor
|
| 28.
|
AG-213
|
See Product Details
|
122520-86-9
|
KI-0311
|
See Product Details
|
| 29.
|
AG-538
|
See Product Details
|
No CAS
|
KI-0312
|
See Product Details
|
| 30.
|
AG-556
|
See Product Details
|
133550-41-1
|
KI-0313
|
See Product Details
|
| 31.
|
Aloisine
|
See Product Details
|
496864-15-4
|
KI-0118
|
Inhibitor of Cdk1/B, Cdk5/p35 and GSK3
|
| 32.
|
AMG-706
|
Not Applicable
|
No CAS
|
KI-0314
|
See Product Details
|
| 33.
|
AMG-TIE2
|
Not Applicable
|
No CAS
|
KI-00585
|
Renal cell carcinoma
|
| 34.
|
Aminogenistein
|
4'-Amino-6-Hydroxyflavone
|
132018-32-7
|
KI-0247
|
Protein tyrosine kinase activity of p561ck
|
| 35.
|
Aminopurvalanol A
|
See Product Details
|
220792-57-4
|
KI-0119
|
CDK & cyclin inhibitors
|
| 36.
|
Apigenin
|
4',5,7-Trihydroxyflavone
|
520-36-5
|
KI-0150
|
Inhibitors of ERK-1/2 proteins
|
| 37.
|
Arctigenin
|
See Product Details
|
7770-78-7
|
KI-0228
|
See Product Details
|
| 38.
|
ARQ-197
|
Not Applicable
|
No CAS
|
KI-00602
|
Breast Cancer
|
| 39.
|
Arqubraf
|
Not Applicable
|
No CAS
|
KI-00603
|
Not Applicable
|
| 40.
|
ARRY-797
|
Not Applicable
|
No CAS
|
KI-00604
|
Glioblastoma multiforme
|
| 41.
|
AS-602801
|
Not Applicable
|
No CAS
|
KI-0315
|
JunKinase inhibitor
|
| 42.
|
AT-7519
|
Not Applicable
|
902135-91-5
|
KI-00580
|
Haematological malignancies
|
| 43.
|
Axitinib
|
AG-013736
|
319460-85-0
|
KI-0087
|
See Product Details
|
| 44.
|
AZ-960
|
Not Applicable
|
No CAS
|
KI-00586
|
Thrombocythemia
|
| 45.
|
AZD-0530
|
Not Applicable
|
No CAS
|
KI-0505
|
See Product Details
|
| 46.
|
AZD-5438
|
Not Applicable
|
No CAS
|
KI-0123
|
Cyclin-dependant kinase (CDK) inhibitor
|
| 47.
|
AZD-6244
|
Not Applicable
|
606143-52-6
|
KI-00576
|
Melanoma
|
| 48.
|
AZD-6703
|
Not Applicable
|
No CAS
|
KI-0316
|
P38 kinase inhibitor
|
| 49.
|
AZD-7762
|
Not Applicable
|
No CAS
|
KI-0317
|
Checkpoint kinase inhibitor
|
| 50.
|
AZM-475271
|
Not Applicable
|
No CAS
|
KI-00605
|
Metastatic bone disease
|
| 51.
|
BAY 61-3606
|
Not Applicable
|
No CAS
|
KI-0441
|
Spleen tyrosine kinase (SYK) inhibitor
|
| 52.
|
BE-23372M
|
Not Applicable
|
No CAS
|
KI-0318
|
Epidermal growth factor (EGF) receptor kinase
|
| 53.
|
BIBU 1361 Dihydrochloride
|
Not Applicable
|
793726-84-8
|
KI-0442
|
See Product Details
|
| 54.
|
BIBW-2992
|
Not Applicable
|
439081-18-2
|
KI-0443
|
EGFR/HER2 tyrosine kinase inhibitor
|
| 55.
|
BI-D1870
|
Not Applicable
|
No CAS
|
KI-0319
|
Inhibits RSK1, RSK2, RSK3 and RSK4
|
| 56.
|
Bisindolylmaleimide (I) Hydrochloride
|
Not Applicable
|
No CAS
|
KI-0208
|
Protein kinase C inhibitors
|
| 57.
|
Bisindolylmaleimide (IX)
|
Not Applicable
|
No CAS
|
KI-0212
|
Protein kinase C inhibitors
|
| 58.
|
Bisindolylmaleimide I
|
See Product Details
|
133052-90-1
|
KI-0207
|
Protein kinase C inhibitors
|
| 59.
|
Bisindolylmaleimide III
|
Not Applicable
|
No CAS
|
KI-0210
|
Protein kinase C inhibitors
|
| 60.
|
Bisindolylmaleimide IV
|
See Product Details
|
119139-23-0
|
KI-0211
|
Protein kinase C inhibitors
|
| 61.
|
Bisindolylmaleimide VI
|
Not Applicable
|
No CAS
|
KI-0213
|
Protein kinase C inhibitors
|
| 62.
|
Bisindolylmaleimide X, Hydrochloride Salt
|
Not Applicable
|
No CAS
|
KI-0214
|
Protein kinase C inhibitors
|
| 63.
|
Bisindolylmaleimide XI, Hydrochloride Salt
|
Not Applicable
|
No CAS
|
KI-0215
|
Protein kinase C inhibitors
|
| 64.
|
BMS-345541
|
Not Applicable
|
547757-23-3
|
KI-0444
|
IKB kinase (IKK) allosteric site inhibitor
|
| 65.
|
BMS-387032
|
See Product Details
|
345627-80-7
|
KI-0482
|
Cyclin dependent kinase (CDK) 2 inhibitor
|
| 66.
|
BMS-536924
|
1H-Benzoimidazol-2-yl)-1H-pyridin-2-one
|
No CAS
|
KI-0019
|
Inhibitor of insulin-like growth factor 1 receptor kinase
|
| 67.
|
BMS-540215
|
Not Applicable
|
649735-46-6
|
KI-0320
|
See Product Details
|
| 68.
|
BMS-582664
|
Brivanib Alaninate
|
No CAS
|
KI-0321
|
Dual inhibitor of VEGFR and FGFR tyrosine kinases
|
| 69.
|
Brivanib
|
BMS-52664
|
No CAS
|
KI-00606
|
Chronic obstructive pulmonary disease
|
| 70.
|
BTK Inhibitor
|
Not Applicable
|
936563-87-0
|
KI-0502
|
Bruton's tyrosine kinase (BTK) inhibitors
|
| 71.
|
Calphostin C
|
Not Applicable
|
121263-19-2
|
KI-0166
|
Inhibitor of protein kinase C
|
| 72.
|
CC-401
|
Not Applicable
|
No CAS
|
KI-0047
|
See Product Details
|
| 73.
|
CEP-1347
|
Not Applicable
|
No CAS
|
KI-0048
|
C-jun amino-terminal kinases (JNKs) inhibitors
|
| 74.
|
CEP-5214
|
Not Applicable
|
No CAS
|
KI-0083
|
Pan-VEGFR tyrosine kinase inhibitor
|
| 75.
|
CEP-701
|
Lestaurtinib
|
111358-88-4
|
KI-0031
|
Inhibitors of FMS-like tyrosine kinase 3 (FLT3)
|
| 76.
|
CEP-7055
|
Not Applicable
|
No CAS
|
KI-0324
|
Pan-VEGFR kinase inhibitor
|
| 77.
|
CGP-53716
|
Not Applicable
|
No CAS
|
KI-0325
|
Tyrosine kinase inhibitor
|
| 78.
|
CGP-57380
|
See Product Details
|
522629-08-9
|
KI-0445
|
See Product Details
|
| 79.
|
CGP-62706
|
Not Applicable
|
No CAS
|
KI-0326
|
Inhibitor of EGF-receptor tyrosine kinase
|
| 80.
|
CGP-74514A Hydrochloride
|
See Product Details
|
No CAS
|
KI-0327
|
Cyclin-dependant kinase-1 (CDK1) inhibitor
|
| 81.
|
CGP-79787 Dihydrochloride
|
See Product Details
|
No CAS
|
KI-0329
|
See Product Details
|
| 82.
|
Chelerythrine Chloride
|
See Product Details
|
3895-92-9
|
KI-0216
|
Selective protein kinase C inhibitor
|
| 83.
|
CHIR-200131
|
Not Applicable
|
No CAS
|
KI-0330
|
RTK inhibitor
|
| 84.
|
CHIR-265
|
Not Applicable
|
No CAS
|
KI-0446
|
Inhibits RAF kinases
|
| 85.
|
CI-1033
|
Not Applicable
|
289499-45-2
|
KI-0135
|
The HER family tyrosine kinase inhibitor
|
| 86.
|
CL-387,785
|
See Product Details
|
No CAS
|
KI-0136
|
Inhibits EGF-receptor (EGFR) kinase
|
| 87.
|
CMPD-1
|
See Product Details
|
41179-33-3
|
KI-0185
|
See Product Details
|
| 88.
|
CNS-9
|
Not Applicable
|
No CAS
|
KI-0332
|
Inhibitor of ABL tyrosine kinase
|
| 89.
|
CP-292597
|
See Product Details
|
No CAS
|
KI-0333
|
See Product Details
|
| 90.
|
CP-673451
|
Not Applicable
|
No CAS
|
KI-0334
|
See Product Details
|
| 91.
|
CP-724714
|
Not Applicable
|
No CAS
|
KI-0026
|
ERBB receptor tyrosine kinase inhibitors
|
| 92.
|
CP-868596
|
Not Applicable
|
No CAS
|
KI-0335
|
See Product Details
|
| 93.
|
CT-53608
|
Not Applicable
|
No CAS
|
KI-0337
|
Inhibitor of FLT-3, PDGFR and C-K
|
| 94.
|
D-4476
|
See Product Details
|
No CAS
|
KI-0509
|
Inhibitor of CK1 (casein kinase 1)
|
| 95
|
Damnacanthal
|
See Product Details
|
477-84-9
|
KI-0222
|
Inhibitor of P56ICK tyrosine kinase 1
|
| 96
|
DMAT
|
2-Dimethylamino-4,5,6,7-tetrabromo-1H-benximidazole
|
No CAS
|
KI-0131
|
CK2 inhibitor
|
| 97
|
DMNB
|
4,5-Dimethoxy-2-nitrobenzaldehyde
|
20357-25-9
|
KI-0134
|
Inhibitor of DNA-dependant protein kinase (DNA-PK)
|
| 98.
|
DMPQ Dihydrochloride
|
5,7-Dimethoxy-3-(4-pyridinyl) quinoline dihydrochloride
|
137206-97-4
|
KI-0272
|
See Product Details
|
| 99.
|
ER-203492-00
|
Not Applicable
|
No CAS
|
KI-0340
|
KDR/FLK-1 tyrosine kinase inhibitor
|
| 100.
|
Erbastatin Analog
|
Methyl 2,5-dihydroxycinnamate
|
63177-57-1
|
KI-0271
|
Inhibits tyrosine kinase
|